.Pharmacolibrary.Drugs.V_Various.V09I_TumourDetection.V09IA10_Technetium99mtcTrofolast.Technetium99mtcTrofolast

Information

name: Technetium99mtcTrofolastatChloride
ATC code: V09IA10
route: intravenous
compartments: 2
dosage: 20 mg
volume of distribution: 15 L
clearance: 1.2 liter/hour
other parameters in model implementation

Technetium (99mTc)trofolastat chloride is a radiopharmaceutical agent used for single-photon emission computed tomography (SPECT) imaging. It functions as a small-molecule inhibitor that binds to prostate-specific membrane antigen (PSMA), a protein often overexpressed in prostate cancer cells. This compound is primarily used in the imaging of prostate cancer for diagnostic purposes. It is not an approved therapeutic drug, but has been used in clinical trials and diagnostic studies.

Pharmacokinetics

Estimated pharmacokinetic parameters for healthy adult males, based primarily on known general PK properties of technetium-99m radiopharmaceuticals, as explicit published PK parameters for technetium (99mTc)trofolastat chloride could not be identified.

References

Revisions


Generated at 2026-04-15T18:18:36Z by OpenModelicaOpenModelica 1.26.3 using GenerateDoc.mos